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Receptor Antagonist
Receptor antagonist
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NMDA receptor antagonists
Nmda receptor antagonist
8a-Phenyld- ecahydroquinoline
MK 801
H2 receptor antagonists
(10)
Famotidine
H2-receptor antagonist
Nizatidine
Burimamide
Cimetidine
Cimetidine
Lafutidine
Metiamide
Pepcid Complete
Ranitidine
Roxatidine
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CB1 receptor antagonists
(11)
AM251
Cannabinoid receptor antagonist
SR141716A
Ibipinabant
LY-320,135
LY-320,135
MK-9470
NESS-0327
Surinabant
Taranabant
Tetrahydro- cannabivarin
VCHSR
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H3 receptor antagonists
ABT-239
Thioperamide
A-423,579
Receptor antagonists
(13)
Endothelin receptor antagonists
Serotonin antagonists
Alpha blockers
Antagonism (chemistry)
Anticholinergics
Anticholinergics
Antihistamines
Beta blockers
CB1 receptor antagonists
GABA antagonists
Kainate receptor antagonists
NMDA receptor antagonists
Opioid antagonist
Tachykinin receptor antagonists
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Signal transduction
Receptors
5-HT
5-HT2A receptor
Opioid receptor
5-HT1 receptor
Histamine receptor
Ligands
Pharmacology
(13)
Dopamine receptor antagonist
B-receptor antagonist
Inverse agonist
Receptor agonist
Competitive antagonist
Competitive antagonist
Lecozotan
Zafirlukast
Radioligand
8a-Phenyld- ecahydroquinoline
ABT-239
Thioperamide
AM251
A-423,579
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5-HT3 antagonists
5-HT3 receptor antagonist
Zatosetron
Bemesetron
Serotonin antagonists
(49)
5-I-R91150
AR-A000002
BRL-15572
SB-216,641
5-HT2A antagonists
5-HT2A antagonists
5-HT2C antagonists
5-HT3 antagonists
9-Aminomet- hyl-9,10-dihydroanthracene
Altanserin
Blonanserin
Cianopramine
Cinanserin
Cyanopindolol
Cyproheptadine
Deramciclane
Dotarizine
EGIS-12233
Eltoprazine
GR-127,935
Iodocyanopindolol
Isamoltane
Ketanserin
LY-272,015
Lecozotan
Lubazodone
Metitepine
Mianserin
NAN-190
Piboserod
Pizotifen
RS-102,221
RS-127,445
Ricasetron
Ritanserin
Ro04-6790
SB-204,741
SB-215,505
SB-242,084
SB-258,585
SB-269,970
SB-271,046
SB-357,134
SB-399,885
SB-699,551
SDZ SER-082
Sarpogrelate
Serotonin antagonist
Trazodone
UH-301
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Transmembrane receptors
(13)
Histamine H2 receptor
D2 receptor
AT1 receptor
CysLT1
5-HT2C receptor
5-HT2C receptor
D1 receptor
Histamine H1 receptor
5-HT2B receptor
5-HT1D receptor
5-HT1B receptor
Glutamate receptor
5-HT4 receptor
Endothelin receptor
more...
Neurotransmitters
(50)
5-HT3 receptor
Dopamine
NMDA
Neuropeptides
Opioids
Opioids
2-Arachido- noylglycerol
5-HT
Acetylcholine
Amino acid neurotransmitter
Anandamide
Aspartic acid
Beta-endorphin
Catecholamine
Cholinergic crisis
Dopaminergic
Dynorphin
Endorphin
Epinephrine
FMRFamide
Gamma-Aminobutyric acid
Gamma-Hydr- oxybutyric acid
Ganglion type nicotinic receptor
Gasotransmitter
Gastrin releasing peptide
Gliotransmitter
Glutamate carboxypeptidase II
Glutamate receptor
Glutamic acid
Glycine
HTR3A
HTR3B
HTR3C
HTR3D
HTR3E
Indirect agonist
Indolamines
Monoamine neurotransmitter
Neurotransmitter
Neurotransmitter transporters
Nitric oxide
Non-noradrenergic, non-cholinergic transmitter
Norepinephrine
Oxytocin
Prodynorphin
Reuptake
Serotonergic
Substance P
Tachykinin peptides
Trace amine
Vasopressin
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Ionotropic receptors
(22)
Ampa receptor
Serotonin receptor
5-HT3 receptor
Cys-loop receptors
GABA receptor
GABA receptor
GRIN1
GRIN3A
GRIN3B
GRINL1A
GRINL1B
Ganglion type nicotinic receptor
Glycine receptor
HTR3A
HTR3B
HTR3C
HTR3D
HTR3E
Kainate receptor
Ligand-gated ion channel
Nicotinic acetylcholine receptor
Nmda receptor
P2X purinoreceptor
more...
Molecular formulas
WAY-100,635
Sulpiride
Orphanin FQ
SCH 23390
BRL-15572
G protein coupled receptors
(26)
Cannabinoid receptor
5-HT1A receptor
Histamine H3 receptor
CB1 receptor
Dopamine receptor
Dopamine receptor
Angiotensin II receptor
Histamine H2 receptor
D2 receptor
AT1 receptor
5-HT2A receptor
Serotonin receptor
CysLT1
Opioid receptor
5-HT2C receptor
D1 receptor
Histamine H1 receptor
5-HT2B receptor
5-HT1D receptor
5-HT1B receptor
Delta opioid receptor
5-HT1 receptor
Muscarinic
Histamine receptor
5-HT4 receptor
Thrombin receptor
Endothelin receptor
more...
Hypothalamic / pituitary axes
(9)
Aldosterone antagonist
Antiandrogen
Antithyroid agent
Corticotropin releasing hormone antagonist
Gonadotrop- in-releasing hormone antagonist
Gonadotrop- in-releasing hormone antagonist
Hypothalam- ic-pituitary-adrenal axis
Hypothalam- ic-pituitary-gonadal axis
Hypothalam- ic-pituitary-thyroid axis
Selective estrogen receptor modulator
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See also
(20)
Leukotriene receptor antagonist
Interleukin 1 receptor antagonist
Angiotensin II receptor antagonist
Angiotensin II receptor antagonists
Endothelin receptor antagonist
Endothelin receptor antagonist
Muscarinic receptor antagonist
H1-receptor antagonist
NK1 receptor antagonist
Beta-receptor antagonist
The Antagonists
Nmda receptor
Sensory receptor
Leukotriene d4
Histamine
Mu opioid receptor
2-Methyl-6- -(phenylethynyl)pyridine
Br J Pharmacol
5-Fluorowillardiine
5-Iodowillardiine
Receptor agonists
more...
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