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CYP3A4
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EC 1.14.14
CYP2D6
CYP2E1
CYP3A
Alkanal monooxygenase (FMN-linked)
Alkanesulfonate monooxygenase
Aromatase
Unspecific monooxygenase
Cytochrome P450
(23)
CYP1A1
CYP1A2
CYP2A6
CYP2B6
CYP2C19
CYP2C19
CYP2C8
CYP2C9
CYP3A7
21-Hydroxylase
Aldosterone synthase
Aromatase
CYP17A1
CYP1B1
CYP27A1
CYP2C9*13
CYP2C9*3
CYP2D6
CYP2E1
CYP3A
Cholesterol side-chain cleavage enzyme
Cytochrome P450 reductase
Lanosterol 14 alpha-demethylase
P450-containing systems
more...
Pharmacokinetics
(30)
ADME-Tox
Drug metabolism
Oral bioavailability
Absorption (pharmacokinetics)
Binding potential
Binding potential
Bioequivalence
Biological half-life
Blood-brain barrier
Clearance (medicine)
Compartment (pharmacokinetics)
Cytochrome p450
Distribution (pharmacology)
Drug action
Enzyme induction and inhibition
First pass effect
Flip-flop kinetics
Free fraction
Haber's Law
Initial volume of distribution
Magnetic marker monitoring
Microdosing
NONMEM
Pharmacokinetics (Population pharmacokinetics)
Physiologi- cally-based pharmacokinetic modelling
Plasma protein binding
Simcyp Simulator
Table of medication secernated in kidney
Table of volume of distribution for drugs
Therapeutic drug monitoring
Volume of distribution
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Metabolism
Xenobiotic
Cytochrome p450
Drug metabolism
Muscarinic antagonists
Solifenacin
Darifenacin
Anti-muscarinic
NK1 receptor antagonists
Aprepitant
Fosaprepitant
Casopitant
L-733,060
NK1 receptor antagonist
Vestipitant
Piperazines
Ketoconazole
Itraconazole
Imatinib mesylate
Indinavir
Aripiprazole
Molecular formulas
(17)
Saquinavir
Pimozide
Cisapride
Ritonavir
Midazolam
Midazolam
Rifampin
Nefazodone
Rifabutin
Alfentanil
Clarithromycin
Amprenavir
Dihydroxyb- ergamottin
Ketoconazole
Itraconazole
Imatinib mesylate
Indinavir
Aripiprazole
more...
Antineoplastic drugs
Nilotinib
Vinorelbine
Temsirolimus
Imatinib mesylate
Protease inhibitors
(19)
Amprenavir
Atazanavir
Boceprevir
Brecanavir
Darunavir
Darunavir
Fosamprenavir
Indinavir
Leupeptin
Lopinavir
Metalloprotease inhibitor
Nelfinavir
Potato carboxypeptidase inhibitor
Protease inhibitor (biology)
Ritonavir
Saquinavir
Secretory leukocyte protease inhibitor
Telaprevir
Tipranavir
Ulinastatin
more...
Cardiac electrophysiology
Qt interval
Torsade de pointes
Antiarrhythmics
QT prolongation
Rifamycin antibiotics
Rifamycin
Rifabutin
Rifampin
Rifapentine
Rifaximin
Proteins
Receptors
Hydroxylation
Isoforms
CYP3A
Gene
PXR
CYP3A5
CYP3A43
CYP2J2
CYP3A4 ligands
Macrolide
PDE5 inhibitor
Ziprasidone
See also
(20)
P-glycoprotein
Eplerenone
Emetogenic
CYP2D6 inhibitors
Concurrent use
Concurrent use
Hepatic
Contraindicated
Microsomes
CYPS
Isoenzyme
Ergotism
Ergot alkaloids
Benzodiazepines
Triazolam
Terfenadine
Carbamazepine
Quinidine
List of drugs affected by grapefruit
Astemizole
Erythromycin breath test
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