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5-ht3 Antagonists
5-HT3 antagonists
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Serotonin antagonists
(48)
5-I-R91150
AR-A000002
BRL-15572
Lecozotan
SB-216,641
SB-216,641
5-HT2A antagonists
5-HT2C antagonists
9-Aminomet- hyl-9,10-dihydroanthracene
Altanserin
Blonanserin
Cianopramine
Cinanserin
Cyanopindolol
Cyproheptadine
Deramciclane
Dotarizine
EGIS-12233
Eltoprazine
GR-127,935
Iodocyanopindolol
Isamoltane
Ketanserin
LY-272,015
Lubazodone
Metitepine
Mianserin
NAN-190
Piboserod
Pizotifen
RS-102,221
RS-127,445
Ricasetron
Ritanserin
Ro04-6790
SB-204,741
SB-215,505
SB-242,084
SB-258,585
SB-269,970
SB-271,046
SB-357,134
SB-399,885
SB-699,551
SDZ SER-082
Sarpogrelate
Serotonin antagonist
Trazodone
UH-301
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Antiemetics
(42)
Antiemetic
Anzemet
Aprepitant
Azasetron
Casopitant
Casopitant
Fosaprepitant
Granisetron
Marinol
Metoclopramide
Metopimazine
Ondansetron
Prochlorperazine
Ramosetron
Tropisetron
5-HT3 antagonist
AS-8112
Acepromazine
Alimemazine
Alizapride
Bendectin
Bromopride
Chlorpromazine
Clebopride
Cyclizine
Dimenhydrinate
Diphenhydramine
Domperidone
Doxylamine
Droperidol
Emetrol
Fluphenazine
Haloperidol
Levomepromazine
Lorazepam
Meclizine
Medical cannabis
Migraleve
Mirtazapine
Nonabine
Paracetamo- l/metoclopramide
Promethazine
Trimethobenzamide
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5-HT3 antagonists
(18)
Alosetron
Bemesetron
Cilansetron
Lerisetron
Palonosetron
Palonosetron
Renzapride
Zacopride
Zatosetron
5-HT3 antagonist
AS-8112
Anzemet
Azasetron
Discovery and development of serotonin receptor antagonists
Granisetron
Lurosetron
Ondansetron
Ramosetron
Tropisetron
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Ionotropic receptors
(22)
5-HT3 receptor
HTR3A
HTR3B
HTR3C
HTR3E
HTR3E
Serotonin receptor
AMPA receptor
Cys-loop receptors
GABA receptor
GRIN1
GRIN3A
GRIN3B
GRINL1A
GRINL1B
Ganglion type nicotinic receptor
Glycine receptor
HTR3D
Kainate receptor
Ligand-gated ion channel
NMDA receptor
Nicotinic acetylcholine receptor
P2X purinoreceptor
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Neurotransmitters
(50)
5-HT
Anandamide
NMDA
Serotonergic
Substance p
Substance p
2-Arachido- noylglycerol
5-HT3 receptor
Acetylcholine
Amino acid neurotransmitter
Aspartic acid
Beta-endorphin
Catecholamine
Cholinergic crisis
Dopamine
Dopaminergic
Dynorphin
Endorphin
Epinephrine
FMRFamide
Gamma-Aminobutyric acid
Gamma-Hydr- oxybutyric acid
Ganglion type nicotinic receptor
Gasotransmitter
Gastrin releasing peptide
Gliotransmitter
Glutamate carboxypeptidase II
Glutamate receptor
Glutamic acid
Glycine
HTR3A
HTR3B
HTR3C
HTR3D
HTR3E
Indirect agonist
Indolamines
Monoamine neurotransmitter
Neuropeptides
Neurotransmitter
Neurotransmitter transporters
Nitric oxide
Non-noradrenergic, non-cholinergic transmitter
Norepinephrine
Opioids
Oxytocin
Prodynorphin
Reuptake
Tachykinin peptides
Trace amine
Vasopressin
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Cell signaling
Receptors
G protein coupled receptors
Autoreceptors
5-HT1 receptor
Presynaptic
5-HT
Signal transduction
(8)
5-HT2A receptor
Receptor antagonist
Receptors
5-HT
G protein coupled receptors
G protein coupled receptors
Autoreceptors
5-HT1 receptor
Presynaptic
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Vomiting
(11)
Emetic
PONV
Antiemetics
Coffee ground vomiting
Cyclic vomiting syndrome
Cyclic vomiting syndrome
Emetophilia
Emetophobia
Hematemesis
Mr Creosote
Retching
Vomiting (Unusual types)
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NK1 receptor antagonists
Neurokinin-1 receptor antagonist
Aprepitant
Casopitant
Fosaprepitant
L-733,060
Vestipitant
G protein coupled receptors
(12)
5-HT1A receptor
5-HT4
5-HT1B receptor
5-HT2C receptor
5-HT2B receptor
5-HT2B receptor
5-HT1D receptor
D2 receptor
5-HT6
Dopamine receptors
Serotonin receptor
5-HT2A receptor
5-HT1 receptor
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Motility stimulants
(12)
Prokinetic
Tegaserod
Alizapride
Bromopride
Cisapride
Cisapride
Clebopride
Domperidone
Itopride
Mebeverine
Metoclopramide
Mosapride
Prucalopride
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Pharmacology
(8)
Cerium oxalate
Locomotor activity
Inverse agonists
Macrogol
Receptor antagonist
Receptor antagonist
Metopimazine
Lecozotan
Azasetron
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See also
(20)
Receptor antagonists
Anatomy
Chemothera- py-induced nausea and vomiting
Dexamethasone
Mesylate
Mesylate
Xylamidine
CYP1A2
Hypromellose
Ventral tegmental area
Gastroparesis
Mesolimbic
Nociceptive
Chemotherapeutic agents
Polysorbate
WAY-100,635
Enterochromaffin cells
Microdialysis
Cisplatin
Glycolate
Cholecystokinin
more...
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