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5-ht3 Antagonist
5-HT3 antagonist
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5-HT3 antagonists
(17)
Alosetron
Anzemet
Azasetron
Bemesetron
Cilansetron
Cilansetron
Granisetron
Lerisetron
Ondansetron
Palonosetron
Ramosetron
Renzapride
Tropisetron
Zacopride
Zatosetron
AS-8112
Discovery and development of serotonin receptor antagonists
Lurosetron
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Antiemetics
(42)
Antiemetic
Aprepitant
Casopitant
Droperidol
Fosaprepitant
Fosaprepitant
Metoclopramide
Metopimazine
Mirtazapine
Prochlorperazine
5-HT3 antagonists
AS-8112
Acepromazine
Alimemazine
Alizapride
Anzemet
Azasetron
Bendectin
Bromopride
Chlorpromazine
Clebopride
Cyclizine
Dimenhydrinate
Diphenhydramine
Domperidone
Doxylamine
Emetrol
Fluphenazine
Granisetron
Haloperidol
Levomepromazine
Lorazepam
Meclizine
Medical cannabis
Migraleve
Nonabine
Ondansetron
Paracetamo- l/metoclopramide
Promethazine
Ramosetron
Tetrahydro- cannabinol
Trimethobenzamide
Tropisetron
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Neurochemistry
Receptor antagonists
Serotonergic
Muscarinic
Ionotropic receptors
(22)
5-HT3
HTR3A
HTR3B
Nicotinic acetylcholine receptor
Nmda receptor
Nmda receptor
Serotonin receptor
AMPA receptor
Cys-loop receptors
GABA receptor
GRIN1
GRIN3A
GRIN3B
GRINL1A
GRINL1B
Ganglion type nicotinic receptor
Glycine receptor
HTR3C
HTR3D
HTR3E
Kainate receptor
Ligand-gated ion channel
P2X purinoreceptor
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Neurotransmitters
(50)
5-HT
Noradrenergic
2-Arachido- noylglycerol
5-HT3
Acetylcholine
Acetylcholine
Amino acid neurotransmitter
Anandamide
Aspartic acid
Beta-endorphin
Catecholamine
Cholinergic crisis
Dopamine
Dopaminergic
Dynorphin
Endorphin
Epinephrine
FMRFamide
Gamma-Aminobutyric acid
Gamma-Hydr- oxybutyric acid
Ganglion type nicotinic receptor
Gasotransmitter
Gastrin releasing peptide
Gliotransmitter
Glutamate carboxypeptidase II
Glutamate receptor
Glutamic acid
Glycine
HTR3A
HTR3B
HTR3C
HTR3D
HTR3E
Indirect agonist
Indolamines
Monoamine neurotransmitter
N-methyl-D-aspartic acid
Neuropeptides
Neurotransmitter
Neurotransmitter transporters
Nitric oxide
Non-noradrenergic, non-cholinergic transmitter
Opioids
Oxytocin
Prodynorphin
Reuptake
Serotonergic
Substance P
Tachykinin peptides
Trace amine
Vasopressin
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Ion channels
5-HT3
HTR3A
HTR3B
Nicotinic acetylcholine receptor
Nmda receptor
Cell signaling
(9)
G protein coupled receptors
Receptors
5-HT2
5-HT1
Postsynaptic
Postsynaptic
Autoreceptors
5-HT
Nicotinic acetylcholine receptor
Nmda receptor
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Signal transduction
(9)
Receptor antagonist
5-HT2A receptor
G protein coupled receptors
Receptors
5-HT
5-HT
5-HT2
5-HT1
Postsynaptic
Autoreceptors
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G protein coupled receptors
(15)
5-HT1A receptor
5-HT2C receptor
5-HT1B receptor
5-HT4 receptor
D2 receptor
D2 receptor
5-HT2B receptor
5-HT1D receptor
Adrenoceptor
5-HT6 receptor
Dopamine receptor
Serotonin receptor
5-HT2A receptor
5-HT2
5-HT1
Muscarinic
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NK1 receptor antagonists
Aprepitant
Casopitant
Fosaprepitant
L-733,060
NK1 receptor antagonist
Vestipitant
Organofluorides
Dexamethasone
5-fluorouracil
Aprepitant
Droperidol
Gastroenterology
Emesis
Gastrocolic response
IBS-D
Ischaemic colitis
Motility stimulants
(12)
Prokinetic
Tegaserod
Alizapride
Bromopride
Cisapride
Cisapride
Clebopride
Domperidone
Itopride
Mebeverine
Metoclopramide
Mosapride
Prucalopride
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Serotonin receptor agonists
5-Carboxam- idotryptamine
8-OH-DPAT
Serotonin agonists
Zacopride
Tegaserod
Pharmacology
(9)
Antispasmodics
Investigational product
Partial agonist
Locomotor activity
Inverse agonists
Inverse agonists
Neuropharmacology
Receptor antagonist
Azasetron
Metopimazine
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Cell biology
Enterochromaffin cells
Microdialysis
Histone H1
Autoreceptors
Serotonergic
5-HT4 agonist
Selective serotonin reuptake enhancer
Serotonin antagonist
Serotonin reuptake inhibitor
See also
(20)
Serotonin antagonists
Chemothera- py-induced nausea and vomiting
CYP1A2
PONV
Anatomy
Anatomy
Br J Pharmacol
AR-A000002
SB-216,641
Antagonist
Serotonin transporter
EC 1.14.14
BRL-15572
Ventral tegmental area
Methylened- ioxyphenyl
Cholecystokinin
Cisplatin
Apomorphine
Indol
Nucleus accumbens
2-oxoglutarate
more...
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